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ºK­n¡G¡uCD4+CD25+ regulatory T cells are involved in the prevention of autoimmune diseases and in tumor-induced tolerance. We previously demonstrated in tumor-bearing rodents that one injection of cyclophosphamide could significantly decrease both numbers and suppressive functions of regulatory T cells, facilitating vaccine-induced tumor rejection. In humans, iterative low dosing of cyclophosphamide, referred to as ¡§metronomic¡¨ therapy, has recently been used in patients with advanced chemotherapy resistant cancers with the aim of reducing tumor angiogenesis. Here we show that oral administration of metronomic cyclophosphamide in advanced cancer patients induces a profound and selective reduction of circulating regulatory T cells, associated with a suppression of their inhibitory functions on conventional T cells and NK cells leading to a restoration of peripheral T cell proliferation and innate killing activities. Therefore, metronomic regimen of cyclophosphamide does not only affect tumor angiogenesis but also strongly curtails immunosuppressive regulatory T cells, favoring a better control of tumor progression. Altogether these data support cyclophosphamide regimen as a valuable treatment for reducing tumor-induced immune tolerance before setting to work anticancer immunotherapy.¡v

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"Cancer immune escape is frequently associated with the induction of an inappropriate immune response,

i.e., a response that does not inhibit but perhaps even promotes the tumor. Indeed, increased frequencies of

tumor-infiltrating regulatory T cells (Tregs) are associated with an impaired prognosis in several cancers.

Thus, depletion of Tregs, e.g., by cyclophosphamide, was proposed as a means to boost immune responses to cancer."

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2 ÁC»ÄÆQ½w½Ä¥Í²zÆQ¤ô¡]Phosphate buffered saline¡A²ºÙ¬°PBS¡^¬O¥Íª«¾Ç¬ã¨s¤¤±`¥Îªº½w½Ä²G

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cyclophosphamide

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(¤wÁp±B ¶PÀù¥­ ¼Ú¬wµµ­m¾J) Ibrance( ¤w¶ùµ¹Letrozole)

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9 the median overall survival (OS) was 37.5 months with Ibrance compared with 33.3 months

with Letrozole alone. (¹êÅç²Õ¤¤¦ì¼ÆÁ`¦s¬¡´Á37.5­Ó¤ë ¹ï·Ó²Õ¤¤¦ì¼ÆÁ`¦s¬¡´Á 33.3­Ó¤ë)

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http://www.obipharma.com/index.aspx?lang=eng&fn=news_content&no=11

Clinical Study Design

The Phase 2/3 randomized controlled trial (RCT) was initiated in December, 2010 with an enrollment target of 342 subjects. The study enrolled female subjects with metastatic breast cancer who achieved stable disease (SD), partial response (PR), or complete response (CR) after at least 1 regimen of anticancer therapy. Subjects were randomized to receive either active treatment (OPT‐822/OPT‐821) plus cyclophosphamide or control (PBS) plus cyclophosphamide in a 2:1 allocation.

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